Assay Detail
Functional
CHEMBL3783898
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Agonist activity at human CB2 receptor expressed in CHO cells after 30 mins by [35S]-GTPgammaS binding assay relative to control
2
Total Activities
1
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Identification of Novel GPR55 Modulators Using Cell-Impedance-Based Label-Free Technology.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Emax | 1 | - | - |
| EC50 | 1 | 6.41 | 6.41 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3781953 | — | — | 2 | 6.41 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3781953 | — | EC50 | = | 391.5 | nM | 6.41 |
| CHEMBL3781953 | — | Emax | = | 87.8 | % | - |