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Assay Detail

CHEMBL3810637

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition AChE (unknown origin) using ATCI as substrate assessed as hydrolysis of ATCI after 10 mins measured every 1 min for 10 times
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Acetylcholinesterase (CHEMBL220)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Bioactive Constituents of Glycyrrhiza uralensis (Licorice): Discovery of the Effective Components of a Traditional Herbal Medicine.
Ji S, Li Z, Song W, Wang Y, Liang W, Li K, Tang S, Wang Q, Qiao X, Zhou D, Yu S, Ye M.
J Nat Prod (2016) 79 : 281 -292
PubMed 26841168 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 5.44 6.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL659 GALANTAMINE 4.0 1 6.52
CHEMBL3809337 1 5.00
CHEMBL1929043 LICORICIDIN 1 4.81

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL659 GALANTAMINE IC50 = 300.0 nM 6.52
CHEMBL3809337 IC50 = 9900.0 nM 5.00
CHEMBL1929043 LICORICIDIN IC50 = 15500.0 nM 4.81