Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL3810649

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of tyrosinase (unknown origin) using L-tyrosine as substrate assessed as oxidation of L-tyrosine after 15 mins
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Tyrosinase (CHEMBL1973)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Bioactive Constituents of Glycyrrhiza uralensis (Licorice): Discovery of the Effective Components of a Traditional Herbal Medicine.
Ji S, Li Z, Song W, Wang Y, Liang W, Li K, Tang S, Wang Q, Qiao X, Zhou D, Yu S, Ye M.
J Nat Prod (2016) 79 : 281 -292
PubMed 26841168 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 6.52 6.81

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1563332 GLYASPERIN D 1 6.81
CHEMBL1630857 GLYASPERIN C 1 6.75
CHEMBL150 KAEMPFEROL 1.0 1 6.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1563332 GLYASPERIN D IC50 = 154.0 nM 6.81
CHEMBL1630857 GLYASPERIN C IC50 = 177.0 nM 6.75
CHEMBL150 KAEMPFEROL IC50 = 1000.0 nM 6.00