Assay Detail
Functional
CHEMBL3820733
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiplasmodial activity against chloroquine-sensitive Plasmodium falciparum D6 by NBT assay
24
Total Activities
24
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Plasmodium falciparum |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Pyrimidine-based antimalarials: design strategies and antiplasmodial effects
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 24 | 8.22 | 8.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3818006 | — | — | 1 | 8.22 |
| CHEMBL3819258 | — | — | 1 | 8.22 |
| CHEMBL3819149 | — | — | 1 | 8.22 |
| CHEMBL3819560 | — | — | 1 | 8.22 |
| CHEMBL3819589 | — | — | 1 | 8.22 |
| CHEMBL3819241 | — | — | 1 | 8.22 |
| CHEMBL3819435 | — | — | 1 | 8.22 |
| CHEMBL3817973 | — | — | 1 | 8.22 |
| CHEMBL3818954 | — | — | 1 | 8.22 |
| CHEMBL3819162 | — | — | 1 | 8.22 |
| CHEMBL3818952 | — | — | 1 | 8.22 |
| CHEMBL3817993 | — | — | 1 | 8.22 |
| CHEMBL3818842 | — | — | 1 | 8.22 |
| CHEMBL3819572 | — | — | 1 | 8.22 |
| CHEMBL3116030 | — | — | 1 | 8.22 |
| CHEMBL3818684 | — | — | 1 | 8.22 |
| CHEMBL3819493 | — | — | 1 | 8.22 |
| CHEMBL3819026 | — | — | 1 | 8.22 |
| CHEMBL3819043 | — | — | 1 | 8.22 |
| CHEMBL3818538 | — | — | 1 | 8.22 |
| CHEMBL3819321 | — | — | 1 | 8.22 |
| CHEMBL3116042 | — | — | 1 | 8.22 |
| CHEMBL3819379 | — | — | 1 | 8.22 |
| CHEMBL3819008 | — | — | 1 | 8.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3818006 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3819258 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3819149 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3819560 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3819589 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3819241 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3819435 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3817973 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3818954 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3819162 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3818952 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3817993 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3818842 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3819572 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3116030 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3818684 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3819493 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3819026 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3819043 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3818538 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3819321 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3116042 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3819379 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3819008 | — | IC50 | = | 6.0 | nM | 8.22 |