Assay Detail
Functional
CHEMBL3826679
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human EOL-1 cells by cell titre glo assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | EOL1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Structure-Based Design of an in Vivo Active Selective BRD9 Inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 5.98 | 6.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3823101 | — | — | 1 | 6.10 |
| CHEMBL3823478 | — | — | 1 | 5.85 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3823101 | — | EC50 | = | 800.0 | nM | 6.10 |
| CHEMBL3823478 | — | EC50 | = | 1400.0 | nM | 5.85 |