Assay Detail
Binding
CHEMBL3829633
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of recombinant human ATX using lysophosphatidylcholine as substrate by choline release assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Development of Autotaxin Inhibitors: An Overview of the Patent and Primary Literature.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 6.88 | 6.88 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3828074 | ZIRITAXESTAT | 3.0 | 1 | 6.88 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3828074 | ZIRITAXESTAT | IC50 | = | 131.0 | nM | 6.88 |