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Assay Detail

CHEMBL3854541

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Toxicity
Cytotoxicity against African green monkey Vero cells
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Toxicity
Organism Chlorocebus sabaeus
Cell Type Vero
Confidence 1 — Organism
Curated By Autocuration

Publication

Lovastatin Analogues from the Soil-Derived Fungus Aspergillus sclerotiorum PSU-RSPG178.
Phainuphong P, Rukachaisirikul V, Saithong S, Phongpaichit S, Bowornwiriyapan K, Muanprasat C, Srimaroeng C, Duangjai A, Sakayaroj J.
J Nat Prod (2016) 79 : 1500 -1507
PubMed 27228159 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 5.18 6.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL123 ELLIPTECINE 1 6.00
CHEMBL503 LOVASTATIN 4.0 1 5.66
CHEMBL3946905 1 5.09
CHEMBL3916495 1 5.08
CHEMBL3978069 1 4.84
CHEMBL3986260 1 4.40

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL123 ELLIPTECINE IC50 = 1000.0 nM 6.00
CHEMBL503 LOVASTATIN IC50 = 2200.0 nM 5.66
CHEMBL3946905 IC50 = 8100.0 nM 5.09
CHEMBL3916495 IC50 = 8400.0 nM 5.08
CHEMBL3978069 IC50 = 14500.0 nM 4.84
CHEMBL3986260 IC50 = 40000.0 nM 4.40