Assay Detail
ADMET
CHEMBL3859772
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of pig heart native MDH reporter reaction after 20 to 40 mins by fluorescence based assay
53
Total Activities
53
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Sus scrofa |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Targeting the HSP60/10 chaperonin systems of Trypanosoma brucei as a strategy for treating African sleeping sickness.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 53 | 4.38 | 4.48 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3910488 | — | — | 1 | 4.48 |
| CHEMBL3907505 | — | — | 1 | 4.39 |
| CHEMBL3938421 | — | — | 1 | 4.33 |
| CHEMBL3986320 | — | — | 1 | 4.30 |
| CHEMBL3906378 | — | — | 1 | - |
| CHEMBL3937258 | — | — | 1 | - |
| CHEMBL3933283 | — | — | 1 | - |
| CHEMBL3960743 | — | — | 1 | - |
| CHEMBL3952045 | — | — | 1 | - |
| CHEMBL3924343 | — | — | 1 | - |
| CHEMBL3978029 | — | — | 1 | - |
| CHEMBL830 | EFLORNITHINE | 4.0 | 1 | - |
| CHEMBL290960 | NIFURTIMOX | 4.0 | 1 | - |
| CHEMBL55 | PENTAMIDINE | 4.0 | 1 | - |
| CHEMBL265502 | SURAMIN | 3.0 | 1 | - |
| CHEMBL3903813 | — | — | 1 | - |
| CHEMBL3953543 | — | — | 1 | - |
| CHEMBL3915348 | — | — | 1 | - |
| CHEMBL3899371 | — | — | 1 | - |
| CHEMBL3943318 | — | — | 1 | - |
| CHEMBL3954893 | — | — | 1 | - |
| CHEMBL3966262 | — | — | 1 | - |
| CHEMBL3955935 | — | — | 1 | - |
| CHEMBL3967047 | — | — | 1 | - |
| CHEMBL3928317 | — | — | 1 | - |
| CHEMBL3947198 | — | — | 1 | - |
| CHEMBL3978830 | — | — | 1 | - |
| CHEMBL3919412 | — | — | 1 | - |
| CHEMBL3908434 | — | — | 1 | - |
| CHEMBL3934352 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3910488 | — | IC50 | = | 33000.0 | nM | 4.48 |
| CHEMBL3907505 | — | IC50 | = | 41000.0 | nM | 4.39 |
| CHEMBL3938421 | — | IC50 | = | 47000.0 | nM | 4.33 |
| CHEMBL3986320 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL3903813 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3979736 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3953543 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3937258 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3975456 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3919336 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3947125 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3912547 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3934460 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3980253 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3951335 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3952406 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3924724 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3115908 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3894125 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3894879 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3922861 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3913878 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3904891 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3983712 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3975683 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3942054 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3983061 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3899371 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3934352 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3908434 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3919412 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3978830 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3947198 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3928317 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3967047 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3955935 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3966262 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3954893 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3943318 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL265502 | SURAMIN | IC50 | > | 63000.0 | nM | - |
| CHEMBL3915348 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3906378 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3933283 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3960743 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3952045 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3924343 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL3978029 | — | IC50 | > | 63000.0 | nM | - |
| CHEMBL830 | EFLORNITHINE | IC50 | > | 63000.0 | nM | - |
| CHEMBL290960 | NIFURTIMOX | IC50 | > | 63000.0 | nM | - |
| CHEMBL55 | PENTAMIDINE | IC50 | > | 63000.0 | nM | - |