Assay Detail
Functional
CHEMBL3864069
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Antiviral activity against HRV1A infected in human HeLa cells assessed as reduction in virus-induced cytopathic effect incubated for 3 days by MTT assay
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Human rhinovirus 1A |
| Cell Type | HeLa |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Rational Design of Novel Highly Potent and Selective Phosphatidylinositol 4-Kinase IIIβ (PI4KB) Inhibitors as Broad-Spectrum Antiviral Agents and Tools for Chemical Biology.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 15 | 6.28 | 7.21 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3959713 | — | — | 1 | 7.21 |
| CHEMBL3947384 | — | — | 1 | 7.16 |
| CHEMBL3976651 | — | — | 1 | 7.12 |
| CHEMBL3923414 | — | — | 1 | 6.18 |
| CHEMBL3930509 | — | — | 1 | 6.14 |
| CHEMBL3893537 | — | — | 1 | 6.00 |
| CHEMBL3902513 | — | — | 1 | 5.27 |
| CHEMBL3911522 | — | — | 1 | 5.17 |
| CHEMBL3894217 | — | — | 1 | - |
| CHEMBL3957128 | — | — | 1 | - |
| CHEMBL3929556 | — | — | 1 | - |
| CHEMBL3948449 | — | — | 1 | - |
| CHEMBL3920652 | — | — | 1 | - |
| CHEMBL3939697 | — | — | 1 | - |
| CHEMBL3958915 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3959713 | — | EC50 | = | 62.0 | nM | 7.21 |
| CHEMBL3947384 | — | EC50 | = | 69.0 | nM | 7.16 |
| CHEMBL3976651 | — | EC50 | = | 75.0 | nM | 7.12 |
| CHEMBL3923414 | — | EC50 | = | 655.0 | nM | 6.18 |
| CHEMBL3930509 | — | EC50 | = | 716.0 | nM | 6.14 |
| CHEMBL3893537 | — | EC50 | = | 990.0 | nM | 6.00 |
| CHEMBL3902513 | — | EC50 | = | 5421.0 | nM | 5.27 |
| CHEMBL3911522 | — | EC50 | = | 6756.0 | nM | 5.17 |
| CHEMBL3894217 | — | EC50 | < | 10.0 | nM | - |
| CHEMBL3957128 | — | EC50 | < | 10.0 | nM | - |
| CHEMBL3929556 | — | EC50 | < | 10.0 | nM | - |
| CHEMBL3948449 | — | EC50 | < | 10.0 | nM | - |
| CHEMBL3920652 | — | EC50 | < | 10.0 | nM | - |
| CHEMBL3939697 | — | EC50 | < | 10.0 | nM | - |
| CHEMBL3958915 | — | EC50 | < | 10.0 | nM | - |