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Assay Detail

CHEMBL3865749

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Mycobacterium tuberculosis H37Rv Eis expressed in Escherichia coli BL21(DE3) using Acetyl-CoA as substrate preincubated for 10 mins followed by substrate addition measured every 30 sec for 10 mins
27
Total Activities
27
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Mycobacterium tuberculosis H37Rv
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

N-acetyltransferase Eis (CHEMBL3879870)
Type SINGLE PROTEIN
Organism Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv)

Publication

Discovery and Optimization of Two Eis Inhibitor Families as Kanamycin Adjuvants against Drug-Resistant M. tuberculosis.
Garzan A, Willby MJ, Green KD, Tsodikov OV, Posey JE, Garneau-Tsodikova S.
ACS Med Chem Lett (2016) 7 : 1219 -1221
PubMed 27994767 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 27 6.13 7.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3931070 1 7.82
CHEMBL1410785 1 7.05
CHEMBL3950034 1 6.80
CHEMBL3976122 1 6.60
CHEMBL3960292 1 6.52
CHEMBL3903088 1 6.52
CHEMBL3927142 1 6.48
CHEMBL3905343 1 6.30
CHEMBL3927499 1 6.27
CHEMBL3980494 1 6.22
CHEMBL3915019 1 5.92
CHEMBL1612166 1 5.66
CHEMBL3926253 1 5.54
CHEMBL3958709 1 5.52
CHEMBL3909271 1 5.24
CHEMBL3890216 1 5.06
CHEMBL3899105 1 4.64
CHEMBL3900249 1 -
CHEMBL3971387 1 -
CHEMBL3979506 1 -
CHEMBL3964177 1 -
CHEMBL3891229 1 -
CHEMBL3940094 1 -
CHEMBL1538832 1 -
CHEMBL3952477 1 -
CHEMBL3976851 1 -
CHEMBL1702313 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3931070 IC50 = 15.0 nM 7.82
CHEMBL1410785 IC50 = 90.0 nM 7.05
CHEMBL3950034 IC50 = 160.0 nM 6.80
CHEMBL3976122 IC50 = 250.0 nM 6.60
CHEMBL3960292 IC50 = 300.0 nM 6.52
CHEMBL3903088 IC50 = 300.0 nM 6.52
CHEMBL3927142 IC50 = 330.0 nM 6.48
CHEMBL3905343 IC50 = 500.0 nM 6.30
CHEMBL3927499 IC50 = 540.0 nM 6.27
CHEMBL3980494 IC50 = 600.0 nM 6.22
CHEMBL3915019 IC50 = 1200.0 nM 5.92
CHEMBL1612166 IC50 = 2200.0 nM 5.66
CHEMBL3926253 IC50 = 2900.0 nM 5.54
CHEMBL3958709 IC50 = 3000.0 nM 5.52
CHEMBL3909271 IC50 = 5800.0 nM 5.24
CHEMBL3890216 IC50 = 8700.0 nM 5.06
CHEMBL3899105 IC50 = 23000.0 nM 4.64
CHEMBL3900249 IC50 > 200000.0 nM -
CHEMBL3971387 IC50 > 200000.0 nM -
CHEMBL3979506 IC50 > 200000.0 nM -
CHEMBL3964177 IC50 > 200000.0 nM -
CHEMBL3891229 IC50 > 200000.0 nM -
CHEMBL3940094 IC50 > 200000.0 nM -
CHEMBL1538832 IC50 > 200000.0 nM -
CHEMBL3952477 IC50 > 200000.0 nM -
CHEMBL3976851 IC50 > 200000.0 nM -
CHEMBL1702313 IC50 > 200000.0 nM -