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Assay Detail

CHEMBL3866628

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Functional
Neuroprotective activity in human SH-SY5Y cells assessed as reduction in 6-OHDA-induced cell death measured after 24 hrs by MTT assay
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type SH-SY5Y
Confidence 1 — Organism
Curated By Autocuration

Publication

Chemical Constituents Isolated from the Root Bark of Cudrania tricuspidata and Their Potential Neuroprotective Effects.
Kwon J, Hiep NT, Kim DW, Hong S, Guo Y, Hwang BY, Lee HJ, Mar W, Lee D.
J Nat Prod (2016) 79 : 1938 -1951
PubMed 27420919 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 10 5.05 5.72

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3604316 1 5.72
CHEMBL140 CURCUMIN 3.0 1 5.21
CHEMBL1977780 1 5.14
CHEMBL303846 XANTHYLETIN 1 5.10
CHEMBL448060 ISOIMPERATORIN 1 5.04
CHEMBL3900419 1 5.04
CHEMBL8659 OLEIC ACID 2.0 1 5.02
CHEMBL452242 GLUTINOL 1 4.89
CHEMBL230558 CUDRAFLAVONE A 1 4.81
CHEMBL14193 4-HYDROXYBENZALDEHYDE 1 4.52

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3604316 EC50 = 1900.0 nM 5.72
CHEMBL140 CURCUMIN EC50 = 6200.0 nM 5.21
CHEMBL1977780 EC50 = 7200.0 nM 5.14
CHEMBL303846 XANTHYLETIN EC50 = 8000.0 nM 5.10
CHEMBL448060 ISOIMPERATORIN EC50 = 9200.0 nM 5.04
CHEMBL3900419 EC50 = 9100.0 nM 5.04
CHEMBL8659 OLEIC ACID EC50 = 9500.0 nM 5.02
CHEMBL452242 GLUTINOL EC50 = 12900.0 nM 4.89
CHEMBL230558 CUDRAFLAVONE A EC50 = 15500.0 nM 4.81
CHEMBL14193 4-HYDROXYBENZALDEHYDE EC50 = 30200.0 nM 4.52