Assay Detail
Functional
CHEMBL3880720
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Cytotoxicity against human HR cells assessed as reduction in cell growth after 72 hrs by MTS assay
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HR |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Novel compounds and methods of use thereof
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 20 | 6.46 | 8.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL301318 | — | — | 1 | 8.10 |
| CHEMBL295063 | — | — | 1 | 7.19 |
| CHEMBL48087 | — | — | 1 | 7.11 |
| CHEMBL3961011 | — | — | 1 | 6.89 |
| CHEMBL3908118 | — | — | 1 | 6.58 |
| CHEMBL3962508 | — | — | 1 | 6.54 |
| CHEMBL46222 | — | — | 1 | 6.53 |
| CHEMBL50280 | — | — | 1 | 6.53 |
| CHEMBL3899298 | — | — | 1 | 6.52 |
| CHEMBL48116 | — | — | 1 | 6.50 |
| CHEMBL295694 | — | — | 1 | 6.49 |
| CHEMBL45601 | — | — | 1 | 6.47 |
| CHEMBL3920818 | — | — | 1 | 6.40 |
| CHEMBL46330 | — | — | 1 | 6.34 |
| CHEMBL296654 | — | — | 1 | 6.26 |
| CHEMBL295137 | — | — | 1 | 6.14 |
| CHEMBL3939453 | — | — | 1 | 6.13 |
| CHEMBL3915216 | — | — | 1 | 5.65 |
| CHEMBL3975937 | — | — | 1 | 5.53 |
| CHEMBL3925025 | — | — | 1 | 5.26 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL301318 | — | IC50 | = | 8.0 | nM | 8.10 |
| CHEMBL295063 | — | IC50 | = | 64.0 | nM | 7.19 |
| CHEMBL48087 | — | IC50 | = | 78.0 | nM | 7.11 |
| CHEMBL3961011 | — | IC50 | = | 128.0 | nM | 6.89 |
| CHEMBL3908118 | — | IC50 | = | 266.0 | nM | 6.58 |
| CHEMBL3962508 | — | IC50 | = | 291.0 | nM | 6.54 |
| CHEMBL46222 | — | IC50 | = | 294.0 | nM | 6.53 |
| CHEMBL50280 | — | IC50 | = | 295.0 | nM | 6.53 |
| CHEMBL3899298 | — | IC50 | = | 300.0 | nM | 6.52 |
| CHEMBL48116 | — | IC50 | = | 316.0 | nM | 6.50 |
| CHEMBL295694 | — | IC50 | = | 324.0 | nM | 6.49 |
| CHEMBL45601 | — | IC50 | = | 340.0 | nM | 6.47 |
| CHEMBL3920818 | — | IC50 | = | 396.0 | nM | 6.40 |
| CHEMBL46330 | — | IC50 | = | 453.0 | nM | 6.34 |
| CHEMBL296654 | — | IC50 | = | 552.0 | nM | 6.26 |
| CHEMBL295137 | — | IC50 | = | 721.0 | nM | 6.14 |
| CHEMBL3939453 | — | IC50 | = | 739.0 | nM | 6.13 |
| CHEMBL3915216 | — | IC50 | = | 2250.0 | nM | 5.65 |
| CHEMBL3975937 | — | IC50 | = | 2984.0 | nM | 5.53 |
| CHEMBL3925025 | — | IC50 | = | 5456.0 | nM | 5.26 |