Assay Detail
ADMET
CHEMBL3880936
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human NHP5 cells
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Homo sapiens |
| Cell Type | NHP5 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Isoform Selective HDAC Inhibitors
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.03 | 4.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL389687 | — | — | 1 | 4.10 |
| CHEMBL389688 | — | — | 1 | 4.00 |
| CHEMBL227170 | — | — | 1 | 4.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL389687 | — | IC50 | = | 80000.0 | nM | 4.10 |
| CHEMBL389688 | — | IC50 | = | 100000.0 | nM | 4.00 |
| CHEMBL227170 | — | IC50 | = | 100000.0 | nM | 4.00 |