Assay Detail
Binding
CHEMBL3882756
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human IGF1R kinase domain (M954 to C1367 residues) tri-phosphorylated enzyme form expressed in baculovirus based expression system using poly-EY peptide incubated for 2 hrs by luciferase-luciferin coupled chemiluminescent assay
527
Total Activities
526
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Insulin-like growth factor 1 receptor (CHEMBL1957) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Pyrimidine Derivatives As Kinase Modulators and Method of Use
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 527 | 6.82 | 7.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3939181 | — | — | 1 | 7.30 |
| CHEMBL3952035 | — | — | 1 | 7.30 |
| CHEMBL3902178 | — | — | 1 | 7.30 |
| CHEMBL3917632 | — | — | 1 | 7.30 |
| CHEMBL3959061 | — | — | 1 | 7.30 |
| CHEMBL3946334 | — | — | 1 | 7.30 |
| CHEMBL3982159 | — | — | 1 | 7.30 |
| CHEMBL3973211 | — | — | 1 | 7.30 |
| CHEMBL3950975 | — | — | 1 | 7.30 |
| CHEMBL3932715 | — | — | 1 | 7.30 |
| CHEMBL3901341 | — | — | 1 | 7.30 |
| CHEMBL505965 | — | — | 1 | 7.30 |
| CHEMBL3958115 | — | — | 1 | 7.30 |
| CHEMBL3978191 | — | — | 1 | 7.30 |
| CHEMBL3975695 | — | — | 1 | 7.30 |
| CHEMBL3943198 | — | — | 1 | 7.30 |
| CHEMBL3929343 | — | — | 1 | 7.30 |
| CHEMBL3902925 | — | — | 1 | 7.30 |
| CHEMBL3918901 | — | — | 1 | 7.30 |
| CHEMBL3917366 | — | — | 1 | 7.30 |
| CHEMBL3951175 | — | — | 1 | 7.30 |
| CHEMBL3904363 | — | — | 1 | 7.30 |
| CHEMBL3968200 | — | — | 1 | 7.30 |
| CHEMBL3945764 | — | — | 1 | 7.30 |
| CHEMBL3907121 | — | — | 1 | 7.30 |
| CHEMBL3904364 | — | — | 1 | 7.30 |
| CHEMBL3974639 | — | — | 1 | 7.30 |
| CHEMBL3920843 | — | — | 1 | 7.30 |
| CHEMBL3911118 | — | — | 1 | 7.30 |
| CHEMBL3958377 | — | — | 1 | 7.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3911765 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3895910 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3911864 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3960772 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3931212 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3974700 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3977190 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3915074 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3938067 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3890207 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3892974 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3949569 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3952184 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL464801 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3914391 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3981560 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3979147 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3920473 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3974093 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL464800 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3913201 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3894512 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3904218 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3980577 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3917671 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3964903 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3929760 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3909730 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3951713 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3961573 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3918853 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3924086 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3921369 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3939968 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3937191 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3916535 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3966630 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3902663 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL1241569 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3977623 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3980001 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3917091 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3919836 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3944113 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3965216 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3971432 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3968695 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3910428 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3907622 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3955053 | — | IC50 | = | 50.0 | nM | 7.30 |