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Assay Detail

CHEMBL3882762

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human NCI-H929 cells assessed as cell growth inhibition after 72 hrs by Cell Titre Glo assay
140
Total Activities
140
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type NCI-H929
Confidence 1 — Organism
Curated By Autocuration

Publication

Imidazopyridine Kinase Inhibitors
(2008)

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 140 6.60 6.60

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3942170 1 6.60
CHEMBL3892197 1 6.60
CHEMBL3918216 1 6.60
CHEMBL3957736 1 6.60
CHEMBL3898691 1 6.60
CHEMBL3944498 1 6.60
CHEMBL3940222 1 6.60
CHEMBL3913169 1 6.60
CHEMBL3974124 1 6.60
CHEMBL3983732 1 6.60
CHEMBL3986506 1 6.60
CHEMBL3907857 1 6.60
CHEMBL3968197 1 6.60
CHEMBL3918852 1 6.60
CHEMBL3921580 1 6.60
CHEMBL3893349 1 6.60
CHEMBL3899043 1 6.60
CHEMBL3898780 1 6.60
CHEMBL3952208 1 6.60
CHEMBL3961740 1 6.60
CHEMBL3946116 1 6.60
CHEMBL3968247 1 6.60
CHEMBL3908294 1 6.60
CHEMBL3911054 1 6.60
CHEMBL3917108 1 6.60
CHEMBL3984698 1 6.60
CHEMBL3934864 1 6.60
CHEMBL3937659 1 6.60
CHEMBL3957642 1 6.60
CHEMBL3920487 1 6.60

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3913169 IC50 = 250.0 nM 6.60
CHEMBL3917108 IC50 = 250.0 nM 6.60
CHEMBL3984698 IC50 = 250.0 nM 6.60
CHEMBL3892197 IC50 = 250.0 nM 6.60
CHEMBL3934864 IC50 = 250.0 nM 6.60
CHEMBL3937659 IC50 = 250.0 nM 6.60
CHEMBL3957642 IC50 = 250.0 nM 6.60
CHEMBL3920487 IC50 = 250.0 nM 6.60
CHEMBL3911054 IC50 = 250.0 nM 6.60
CHEMBL3908294 IC50 = 250.0 nM 6.60
CHEMBL3968247 IC50 = 250.0 nM 6.60
CHEMBL3946116 IC50 = 250.0 nM 6.60
CHEMBL3961740 IC50 = 250.0 nM 6.60
CHEMBL3952208 IC50 = 250.0 nM 6.60
CHEMBL3898780 IC50 = 250.0 nM 6.60
CHEMBL3942170 IC50 = 250.0 nM 6.60
CHEMBL3899043 IC50 = 250.0 nM 6.60
CHEMBL3893349 IC50 = 250.0 nM 6.60
CHEMBL3940222 IC50 = 250.0 nM 6.60
CHEMBL3944498 IC50 = 250.0 nM 6.60
CHEMBL3974124 IC50 = 250.0 nM 6.60
CHEMBL3898691 IC50 = 250.0 nM 6.60
CHEMBL3983732 IC50 = 250.0 nM 6.60
CHEMBL3986506 IC50 = 250.0 nM 6.60
CHEMBL3918216 IC50 = 250.0 nM 6.60
CHEMBL3907857 IC50 = 250.0 nM 6.60
CHEMBL3968197 IC50 = 250.0 nM 6.60
CHEMBL3918852 IC50 = 250.0 nM 6.60
CHEMBL3921580 IC50 = 250.0 nM 6.60
CHEMBL3957736 IC50 = 250.0 nM 6.60
CHEMBL3912500 IC50 < 250.0 nM -
CHEMBL3915154 IC50 < 250.0 nM -
CHEMBL3896003 IC50 > 1000.0 nM -
CHEMBL3919927 IC50 < 250.0 nM -
CHEMBL3976565 IC50 < 250.0 nM -
CHEMBL3967372 IC50 < 250.0 nM -
CHEMBL3951411 IC50 < 250.0 nM -
CHEMBL506862 IC50 < 250.0 nM -
CHEMBL3954082 IC50 < 250.0 nM -
CHEMBL3952960 IC50 < 250.0 nM -
CHEMBL3938801 IC50 < 250.0 nM -
CHEMBL3918624 IC50 < 250.0 nM -
CHEMBL3941932 IC50 < 250.0 nM -
CHEMBL3890964 IC50 < 250.0 nM -
CHEMBL3986972 IC50 < 250.0 nM -
CHEMBL3984255 IC50 < 250.0 nM -
CHEMBL3901948 IC50 < 250.0 nM -
CHEMBL3909461 IC50 < 250.0 nM -
CHEMBL3905860 IC50 < 250.0 nM -
CHEMBL3930103 IC50 < 250.0 nM -