Assay Detail
Functional
CHEMBL3883099
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human recombinant EP4 receptor expressed in HEK293 cells assessed as effect on calcium accumulation by Fluo-4 AM dye based FLIPR assay
124
Total Activities
124
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Prostaglandin E2 receptor EP4 subtype (CHEMBL1836) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Therapeutic compounds
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 124 | 4.83 | 5.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3959926 | — | — | 1 | 5.00 |
| CHEMBL3948932 | — | — | 1 | 4.65 |
| CHEMBL3955642 | — | — | 1 | - |
| CHEMBL3967458 | — | — | 1 | - |
| CHEMBL3903558 | — | — | 1 | - |
| CHEMBL3906280 | — | — | 1 | - |
| CHEMBL3949225 | — | — | 1 | - |
| CHEMBL3951834 | — | — | 1 | - |
| CHEMBL3918028 | — | — | 1 | - |
| CHEMBL3920755 | — | — | 1 | - |
| CHEMBL3958410 | — | — | 1 | - |
| CHEMBL3902125 | — | — | 1 | - |
| CHEMBL3899346 | — | — | 1 | - |
| CHEMBL3930718 | — | — | 1 | - |
| CHEMBL3967265 | — | — | 1 | - |
| CHEMBL3915820 | — | — | 1 | - |
| CHEMBL3890808 | — | — | 1 | - |
| CHEMBL3953564 | — | — | 1 | - |
| CHEMBL3963968 | — | — | 1 | - |
| CHEMBL3922332 | — | — | 1 | - |
| CHEMBL3890334 | — | — | 1 | - |
| CHEMBL3982222 | — | — | 1 | - |
| CHEMBL3984757 | — | — | 1 | - |
| CHEMBL3985691 | — | — | 1 | - |
| CHEMBL3968706 | — | — | 1 | - |
| CHEMBL3969714 | — | — | 1 | - |
| CHEMBL3972401 | — | — | 1 | - |
| CHEMBL3937945 | — | — | 1 | - |
| CHEMBL3953958 | — | — | 1 | - |
| CHEMBL3917878 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3959926 | — | EC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL3948932 | — | EC50 | = | 22457.0 | nM | 4.65 |
| CHEMBL3921784 | — | EC50 | - | — | - | |
| CHEMBL3906402 | — | EC50 | - | — | - | |
| CHEMBL3892847 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3947001 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3901873 | — | EC50 | - | — | - | |
| CHEMBL3915040 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3909754 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3938844 | — | EC50 | - | — | - | |
| CHEMBL3973347 | — | EC50 | - | — | - | |
| CHEMBL3936540 | — | EC50 | - | — | - | |
| CHEMBL3959653 | — | EC50 | - | — | - | |
| CHEMBL1722929 | — | EC50 | - | — | - | |
| CHEMBL3922151 | — | EC50 | - | — | - | |
| CHEMBL3920796 | — | EC50 | - | — | - | |
| CHEMBL3918084 | — | EC50 | - | — | - | |
| CHEMBL3903611 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3896863 | — | EC50 | - | — | - | |
| CHEMBL3924461 | — | EC50 | - | — | - | |
| CHEMBL3934163 | — | EC50 | - | — | - | |
| CHEMBL3924999 | — | EC50 | - | — | - | |
| CHEMBL3898377 | — | EC50 | - | — | - | |
| CHEMBL3917796 | — | EC50 | - | — | - | |
| CHEMBL3920521 | — | EC50 | - | — | - | |
| CHEMBL3974000 | — | EC50 | - | — | - | |
| CHEMBL3983069 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3908484 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3905606 | — | EC50 | - | — | - | |
| CHEMBL3908432 | — | EC50 | - | — | - | |
| CHEMBL3935916 | — | EC50 | - | — | - | |
| CHEMBL3945620 | — | EC50 | - | — | - | |
| CHEMBL3936978 | — | EC50 | - | — | - | |
| CHEMBL3934202 | — | EC50 | - | — | - | |
| CHEMBL3973963 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3986923 | — | EC50 | - | — | - | |
| CHEMBL3897181 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3920560 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3920756 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3927083 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3901088 | — | EC50 | - | — | - | |
| CHEMBL3898314 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3922270 | — | EC50 | - | — | - | |
| CHEMBL3924987 | — | EC50 | - | — | - | |
| CHEMBL3975238 | — | EC50 | - | — | - | |
| CHEMBL3977724 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3907809 | — | EC50 | - | — | - | |
| CHEMBL3918349 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3959769 | — | EC50 | - | — | - | |
| CHEMBL3971632 | — | EC50 | > | 10000.0 | nM | - |