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Assay Detail

CHEMBL3998992

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Enterovirus 71 TW/70902/08 clinical isolates incubated for 2 to 3 days
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Enterovirus A71
Confidence 1 — Organism
Curated By Autocuration

Target

Enterovirus A71 (CHEMBL612436)
Type ORGANISM
Organism Enterovirus A71

Publication

Discovery of Multitarget Agents Active as Broad-Spectrum Antivirals and Correctors of Cystic Fibrosis Transmembrane Conductance Regulator for Associated Pulmonary Diseases.
Tassini S, Sun L, Lanko K, Crespan E, Langron E, Falchi F, Kissova M, Armijos-Rivera JI, Delang L, Mirabelli C, Neyts J, Pieroni M, Cavalli A, Costantino G, Maga G, Vergani P, Leyssen P, Radi M.
J Med Chem (2017) 60 : 1400 -1416
PubMed 28122178 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 5.45 5.45

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4085374 1 5.45

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4085374 EC50 = 3580.0 nM 5.45