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Assay Detail

CHEMBL4000328

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Herpes simplex virus 2 G infected in human HEL cells assessed as inhibition of virus-induced cytopathic effect by visual scoring analysis
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human alphaherpesvirus 2
Confidence 1 — Organism
Curated By Autocuration

Target

Human alphaherpesvirus 2 (CHEMBL370)
Type ORGANISM
Organism Human alphaherpesvirus 2

Publication

Synthesis, antiplasmodial activity and mechanistic studies of pyrimidine-5-carbonitrile and quinoline hybrids.
Kaur H, Balzarini J, de Kock C, Smith PJ, Chibale K, Singh K.
Eur J Med Chem (2015) 101 : 52 -62
PubMed 26114811 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 14 7.00 7.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL184 ACYCLOVIR 4.0 1 7.00
CHEMBL4066702 1 -
CHEMBL4088000 1 -
CHEMBL4069858 1 -
CHEMBL4097050 1 -
CHEMBL4080544 1 -
CHEMBL4104770 1 -
CHEMBL4088409 1 -
CHEMBL4067148 1 -
CHEMBL4096132 1 -
CHEMBL4078078 1 -
CHEMBL4083981 1 -
CHEMBL4062263 1 -
CHEMBL76 CHLOROQUINE 4.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL184 ACYCLOVIR EC50 = 100.0 nM 7.00
CHEMBL4066702 EC50 > 4000.0 nM -
CHEMBL4088000 EC50 > 800.0 nM -
CHEMBL4069858 EC50 > 800.0 nM -
CHEMBL4097050 EC50 > 100000.0 nM -
CHEMBL4080544 EC50 > 4000.0 nM -
CHEMBL4104770 EC50 > 800.0 nM -
CHEMBL4088409 EC50 > 100000.0 nM -
CHEMBL4067148 EC50 > 800.0 nM -
CHEMBL4096132 EC50 > 100000.0 nM -
CHEMBL4078078 EC50 > 800.0 nM -
CHEMBL4083981 EC50 > 4000.0 nM -
CHEMBL4062263 EC50 > 4000.0 nM -
CHEMBL76 CHLOROQUINE EC50 > 20000.0 nM -