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Assay Detail

CHEMBL4000421

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Cytotoxicity against mouse L929 cells after 5 days by MTT assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Mus musculus
Cell Type L929
Confidence 1 — Organism
Curated By Autocuration

Target

L929 (CHEMBL612267)
Type CELL-LINE
Organism Mus musculus

Publication

Pyristriatins A and B: Pyridino-Cyathane Antibiotics from the Basidiomycete Cyathus cf. striatus.
Richter C, Helaly SE, Thongbai B, Hyde KD, Stadler M.
J Nat Prod (2016) 79 : 1684 -1688
PubMed 27231731 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 6.01 8.42

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL329993 EPOTHILONE A 1 8.42
CHEMBL4071721 1 4.81
CHEMBL4082991 1 4.79

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL329993 EPOTHILONE A IC50 = 3.8 nM 8.42
CHEMBL4071721 IC50 = 15400.0 nM 4.81
CHEMBL4082991 IC50 = 16300.0 nM 4.79