Assay Detail
Binding
CHEMBL4023938
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Binding affinity to CA7 (unknown origin) assessed as intrinsic thermodynamic equilibrium constant at pH 7 by SPR assay
17
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Introduction of Intrinsic Kinetics of Protein-Ligand Interactions and Their Implications for Drug Design.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 17 | 9.08 | 10.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2011156 | — | — | 1 | 10.68 |
| CHEMBL3797385 | — | — | 1 | 10.42 |
| CHEMBL2443188 | — | — | 1 | 10.00 |
| CHEMBL3799577 | — | — | 1 | 9.77 |
| CHEMBL2333416 | — | — | 1 | 9.72 |
| CHEMBL2010994 | — | — | 1 | 9.64 |
| CHEMBL3798446 | — | — | 1 | 9.48 |
| CHEMBL3797893 | — | — | 1 | 9.18 |
| CHEMBL3359181 | — | — | 1 | 8.77 |
| CHEMBL3799296 | — | — | 1 | 8.68 |
| CHEMBL1272242 | — | — | 1 | 8.62 |
| CHEMBL2011155 | — | — | 1 | 8.44 |
| CHEMBL2443189 | — | — | 1 | 8.41 |
| CHEMBL3359179 | — | — | 1 | 8.31 |
| CHEMBL1272187 | — | — | 1 | 7.89 |
| CHEMBL3799945 | — | — | 1 | 7.23 |
| CHEMBL3798473 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2011156 | — | Kd | = | 0.021 | nM | 10.68 |
| CHEMBL3797385 | — | Kd | = | 0.038 | nM | 10.42 |
| CHEMBL2443188 | — | Kd | = | 0.1 | nM | 10.00 |
| CHEMBL3799577 | — | Kd | = | 0.17 | nM | 9.77 |
| CHEMBL2333416 | — | Kd | = | 0.19 | nM | 9.72 |
| CHEMBL2010994 | — | Kd | = | 0.23 | nM | 9.64 |
| CHEMBL3798446 | — | Kd | = | 0.33 | nM | 9.48 |
| CHEMBL3797893 | — | Kd | = | 0.66 | nM | 9.18 |
| CHEMBL3359181 | — | Kd | = | 1.7 | nM | 8.77 |
| CHEMBL3799296 | — | Kd | = | 2.1 | nM | 8.68 |
| CHEMBL1272242 | — | Kd | = | 2.4 | nM | 8.62 |
| CHEMBL2011155 | — | Kd | = | 3.6 | nM | 8.44 |
| CHEMBL2443189 | — | Kd | = | 3.9 | nM | 8.41 |
| CHEMBL3359179 | — | Kd | = | 4.9 | nM | 8.31 |
| CHEMBL1272187 | — | Kd | = | 13.0 | nM | 7.89 |
| CHEMBL3799945 | — | Kd | = | 59.0 | nM | 7.23 |
| CHEMBL3798473 | — | Kd | = | 0.0041 | nM | - |