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Assay Detail

CHEMBL4024922

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Functional
Cytotoxicity against human LNCAP cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type LNCaP
Confidence 1 — Organism
Curated By Autocuration

Target

LNCaP (CHEMBL612518)
Type CELL-LINE
Organism Homo sapiens

Publication

Identification of highly potent and selective PI3Kδ inhibitors.
Marcoux D, Qin LY, Ruan Z, Shi Q, Ruan Q, Weigelt C, Qiu H, Schieven G, Hynes J, Bhide R, Poss M, Tino J.
Bioorg Med Chem Lett (2017) 27 : 2849 -2853
PubMed 28209465 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.24 5.24

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4091875 1 5.24

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4091875 IC50 = 5700.0 nM 5.24