Assay Detail
Functional
CHEMBL4030956
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Agonist activity at human GPCR41 transfected in HEK293 cells assessed as [35S]GTPgammaS binding by scintillation counting method
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Microbiota-Host Transgenomic Metabolism, Bioactive Molecules from the Inside.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3 | 4.92 | 4.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL14227 | BUTYRIC ACID | 2.0 | 1 | 4.92 |
| CHEMBL14021 | PROPIONIC ACID | 2.0 | 1 | 4.92 |
| CHEMBL539 | ACETIC ACID | 4.0 | 1 | 4.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL14227 | BUTYRIC ACID | EC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL14021 | PROPIONIC ACID | EC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL539 | ACETIC ACID | EC50 | = | 12000.0 | nM | 4.92 |