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Assay Detail

CHEMBL4035575

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [3H]DTG from sigma-2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting method
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Rattus norvegicus
Tissue Liver
Subcellular Membrane
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Sigma intracellular receptor 2 (CHEMBL4105864)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Lipase-catalyzed kinetic resolution as key step in the synthesis of enantiomerically pure σ ligands with 2-benzopyran structure.
Knappmann I, Lehmkuhl K, Köhler J, Schepmann D, Giera M, Bracher F, Wünsch B.
Bioorg Med Chem (2017) 25 : 3384 -3395
PubMed 28501431 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 10 6.67 7.50

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3828752 1 7.50
CHEMBL282433 DITOLYLGUANIDINE 1 7.38
CHEMBL4092162 1 7.17
CHEMBL54 HALOPERIDOL 4.0 1 7.11
CHEMBL4102372 1 6.58
CHEMBL1169963 1 6.29
CHEMBL1171865 1 6.29
CHEMBL4077547 1 6.28
CHEMBL1172685 1 6.21
CHEMBL1169962 1 5.91

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3828752 Ki = 32.0 nM 7.50
CHEMBL282433 DITOLYLGUANIDINE Ki = 42.0 nM 7.38
CHEMBL4092162 Ki = 68.0 nM 7.17
CHEMBL54 HALOPERIDOL Ki = 78.0 nM 7.11
CHEMBL4102372 Ki = 260.0 nM 6.58
CHEMBL1169963 Ki = 519.0 nM 6.29
CHEMBL1171865 Ki = 510.0 nM 6.29
CHEMBL4077547 Ki = 525.0 nM 6.28
CHEMBL1172685 Ki = 614.0 nM 6.21
CHEMBL1169962 Ki = 1220.0 nM 5.91