Assay Detail
Binding
CHEMBL4041970
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of recombinant Leishmania donovani DYRK4 expressed in Escherichia coli using woodtide as substrate after 30 mins in presence of [gamma-33P]ATP by liquid scintillation counting
60
Total Activities
60
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Leishmania donovani |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Exploration of the imidazo[1,2-b]pyridazine scaffold as a protein kinase inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 60 | 5.00 | 5.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4062820 | — | — | 1 | 5.00 |
| CHEMBL4082981 | — | — | 1 | 5.00 |
| CHEMBL4090223 | — | — | 1 | - |
| CHEMBL4072506 | — | — | 1 | - |
| CHEMBL4077125 | — | — | 1 | - |
| CHEMBL4062568 | — | — | 1 | - |
| CHEMBL4067420 | — | — | 1 | - |
| CHEMBL4091127 | — | — | 1 | - |
| CHEMBL4063254 | — | — | 1 | - |
| CHEMBL4098107 | — | — | 1 | - |
| CHEMBL4079347 | — | — | 1 | - |
| CHEMBL4079343 | — | — | 1 | - |
| CHEMBL4076663 | — | — | 1 | - |
| CHEMBL4084919 | — | — | 1 | - |
| CHEMBL4102871 | — | — | 1 | - |
| CHEMBL4062683 | — | — | 1 | - |
| CHEMBL4092117 | — | — | 1 | - |
| CHEMBL4093104 | — | — | 1 | - |
| CHEMBL4065432 | — | — | 1 | - |
| CHEMBL4070227 | — | — | 1 | - |
| CHEMBL4071413 | — | — | 1 | - |
| CHEMBL4098237 | — | — | 1 | - |
| CHEMBL4071322 | — | — | 1 | - |
| CHEMBL4083948 | — | — | 1 | - |
| CHEMBL4075509 | — | — | 1 | - |
| CHEMBL4074499 | — | — | 1 | - |
| CHEMBL4071013 | — | — | 1 | - |
| CHEMBL4064988 | — | — | 1 | - |
| CHEMBL4092673 | — | — | 1 | - |
| CHEMBL4074132 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4062820 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL4082981 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL4062568 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4080844 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4077125 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4072506 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4090223 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4069158 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4100956 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4081668 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4091942 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4076906 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4070065 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4097256 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4061394 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4089542 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4087260 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4076448 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4077159 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4093231 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4075820 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4085467 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4090770 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4084364 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4086402 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4104296 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4065432 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4074132 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4092673 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4064988 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4071013 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4074499 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4075509 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4083948 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4071322 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4098237 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4071413 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4070227 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4067420 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4093104 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4092117 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4062683 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4102871 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4084919 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4076663 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4079343 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4079347 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4098107 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4063254 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4091127 | — | IC50 | > | 10000.0 | nM | - |