Assay Detail
Binding
CHEMBL4044889
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Inhibition of C-terminal biotin-labelled BCoR/wild-type BCL6 BTB domain (unknown origin) protein-protein interaction by ELISA
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Discovery of a novel B-cell lymphoma 6 (BCL6)-corepressor interaction inhibitor by utilizing structure-based drug design.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 19 | 5.73 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4075278 | — | — | 1 | 7.00 |
| CHEMBL4076344 | — | — | 1 | 6.89 |
| CHEMBL4076619 | — | — | 1 | 6.89 |
| CHEMBL4085850 | — | — | 1 | 6.89 |
| CHEMBL4103775 | — | — | 1 | 6.82 |
| CHEMBL4069588 | — | — | 1 | 6.66 |
| CHEMBL4093597 | — | — | 1 | 6.62 |
| CHEMBL4066000 | — | — | 1 | 6.37 |
| CHEMBL4092657 | — | — | 1 | 5.37 |
| CHEMBL4063725 | — | — | 1 | 5.35 |
| CHEMBL4084898 | — | — | 1 | 5.07 |
| CHEMBL4096591 | — | — | 1 | 4.85 |
| CHEMBL4074632 | — | — | 1 | 4.37 |
| CHEMBL4101332 | — | — | 1 | 4.21 |
| CHEMBL1517539 | — | — | 1 | 4.16 |
| CHEMBL4070173 | — | — | 1 | 4.08 |
| CHEMBL4070563 | — | — | 1 | - |
| CHEMBL4063249 | TP-021n | — | 1 | - |
| CHEMBL4066375 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4075278 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL4076344 | — | IC50 | = | 130.0 | nM | 6.89 |
| CHEMBL4076619 | — | IC50 | = | 130.0 | nM | 6.89 |
| CHEMBL4085850 | — | IC50 | = | 130.0 | nM | 6.89 |
| CHEMBL4103775 | — | IC50 | = | 150.0 | nM | 6.82 |
| CHEMBL4069588 | — | IC50 | = | 220.0 | nM | 6.66 |
| CHEMBL4093597 | — | IC50 | = | 240.0 | nM | 6.62 |
| CHEMBL4066000 | — | IC50 | = | 430.0 | nM | 6.37 |
| CHEMBL4092657 | — | IC50 | = | 4300.0 | nM | 5.37 |
| CHEMBL4063725 | — | IC50 | = | 4500.0 | nM | 5.35 |
| CHEMBL4084898 | — | IC50 | = | 8600.0 | nM | 5.07 |
| CHEMBL4096591 | — | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL4074632 | — | IC50 | = | 43000.0 | nM | 4.37 |
| CHEMBL4101332 | — | IC50 | = | 62000.0 | nM | 4.21 |
| CHEMBL1517539 | — | IC50 | = | 69000.0 | nM | 4.16 |
| CHEMBL4070173 | — | IC50 | = | 83000.0 | nM | 4.08 |
| CHEMBL4070563 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL4063249 | TP-021n | IC50 | = | 110000.0 | nM | - |
| CHEMBL4066375 | — | IC50 | = | 200000.0 | nM | - |