Assay Detail
Functional
CHEMBL4047455
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Agonist activity at mouse NMUR1 expressed in CHO cells assessed as increase in intracellular calcium influx after 180 secs by Fluo 4-AM dye based FLIPR assay
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
A potent neuromedin U receptor 2-selective alkylated peptide.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 20 | 7.19 | 9.09 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3356083 | — | — | 1 | 9.09 |
| CHEMBL4074121 | — | — | 1 | 8.02 |
| CHEMBL4097408 | — | — | 1 | 7.23 |
| CHEMBL4081819 | — | — | 1 | 7.17 |
| CHEMBL4103826 | — | — | 1 | 7.16 |
| CHEMBL4088810 | — | — | 1 | 7.12 |
| CHEMBL4073508 | — | — | 1 | 7.10 |
| CHEMBL4079565 | — | — | 1 | 7.03 |
| CHEMBL4076016 | — | — | 1 | 7.00 |
| CHEMBL4094147 | — | — | 1 | 6.96 |
| CHEMBL4080881 | — | — | 1 | 6.96 |
| CHEMBL4071009 | — | — | 1 | 6.77 |
| CHEMBL4070228 | — | — | 1 | 6.54 |
| CHEMBL4105113 | — | — | 1 | 6.52 |
| CHEMBL4092080 | — | — | 1 | - |
| CHEMBL4083670 | — | — | 1 | - |
| CHEMBL4061906 | — | — | 1 | - |
| CHEMBL4060830 | — | — | 1 | - |
| CHEMBL4087316 | — | — | 1 | - |
| CHEMBL4067577 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3356083 | — | EC50 | = | 0.81 | nM | 9.09 |
| CHEMBL4074121 | — | EC50 | = | 9.6 | nM | 8.02 |
| CHEMBL4097408 | — | EC50 | = | 59.0 | nM | 7.23 |
| CHEMBL4081819 | — | EC50 | = | 67.0 | nM | 7.17 |
| CHEMBL4103826 | — | EC50 | = | 70.0 | nM | 7.16 |
| CHEMBL4088810 | — | EC50 | = | 76.0 | nM | 7.12 |
| CHEMBL4073508 | — | EC50 | = | 80.0 | nM | 7.10 |
| CHEMBL4079565 | — | EC50 | = | 94.0 | nM | 7.03 |
| CHEMBL4076016 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL4094147 | — | EC50 | = | 110.0 | nM | 6.96 |
| CHEMBL4080881 | — | EC50 | = | 110.0 | nM | 6.96 |
| CHEMBL4071009 | — | EC50 | = | 170.0 | nM | 6.77 |
| CHEMBL4070228 | — | EC50 | = | 290.0 | nM | 6.54 |
| CHEMBL4105113 | — | EC50 | = | 300.0 | nM | 6.52 |
| CHEMBL4092080 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL4083670 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL4061906 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL4060830 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL4087316 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL4067577 | — | EC50 | > | 1000.0 | nM | - |