Assay Detail
Functional
CHEMBL4049705
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Antiproliferative activity against human HCT116 cells after 72 hrs by Cell Titer-Glo assay
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HCT-116 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Discovery of an Inhibitor of the Proteasome Subunit Rpn11.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 11 | 5.55 | 5.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4076575 | — | — | 1 | 5.80 |
| CHEMBL4101230 | — | — | 1 | 5.68 |
| CHEMBL4100994 | — | — | 1 | 5.58 |
| CHEMBL4084782 | — | — | 1 | 5.47 |
| CHEMBL310555 | OXYQUINOLINE | -1.0 | 1 | 5.22 |
| CHEMBL4094874 | — | — | 1 | - |
| CHEMBL1702610 | — | — | 1 | - |
| CHEMBL4076981 | — | — | 1 | - |
| CHEMBL4075311 | — | — | 1 | - |
| CHEMBL4083010 | — | — | 1 | - |
| CHEMBL4063134 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4076575 | — | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL4101230 | — | IC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL4100994 | — | IC50 | = | 2600.0 | nM | 5.58 |
| CHEMBL4084782 | — | IC50 | = | 3400.0 | nM | 5.47 |
| CHEMBL310555 | OXYQUINOLINE | IC50 | = | 6000.0 | nM | 5.22 |
| CHEMBL4094874 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1702610 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4076981 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4075311 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4083010 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4063134 | — | IC50 | > | 10000.0 | nM | - |