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Assay Detail

CHEMBL4120902

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to recombinant HMGB1 box A (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

High mobility group protein B1 (CHEMBL2311236)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

High Mobility Group Box-1 (HMGb1): Current Wisdom and Advancement as a Potential Drug Target.
VanPatten S, Al-Abed Y.
J Med Chem (2018) 61 : 5093 -5107
PubMed 29268019 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 2 7.42 8.83

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4129393 1 8.83
CHEMBL424 SALICYLIC ACID 3.0 1 6.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4129393 Kd = 1.48 nM 8.83
CHEMBL424 SALICYLIC ACID Kd = 1000.0 nM 6.00