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Assay Detail

CHEMBL4123978

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Binding
Inhibition of Dengue virus 4 NS5 full length RdRp activity using RNA as template assessed as inhibition of NTPs incorporation after 90 mins by FAPA assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism dengue virus type 4
Confidence 8 — Homologous single protein target
Curated By Intermediate

Target

Nonstructural protein 5 (CHEMBL4295629)
Type SINGLE PROTEIN
Organism Dengue virus

Publication

Structure-activity relationship of uridine-based nucleoside phosphoramidate prodrugs for inhibition of dengue virus RNA-dependent RNA polymerase.
Wang G, Lim SP, Chen YL, Hunziker J, Rao R, Gu F, Seh CC, Ghafar NA, Xu H, Chan K, Lin X, Saunders OL, Fenaux M, Zhong W, Shi PY, Yokokawa F.
Bioorg Med Chem Lett (2018) 28 : 2324 -2327
PubMed 29801997 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.47 6.47

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4126343 1 6.47

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4126343 IC50 = 340.0 nM 6.47