Assay Detail
Functional
CHEMBL4124802
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assay
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Gastric inhibitory polypeptide receptor (CHEMBL4383) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Dual Glucagon-like Peptide 1 (GLP-1)/Glucagon Receptor Agonists Specifically Optimized for Multidose Formulations.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 16 | 8.99 | 10.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4127525 | — | — | 1 | 10.40 |
| CHEMBL4126812 | — | — | 1 | 10.24 |
| CHEMBL4129347 | — | — | 1 | 9.99 |
| CHEMBL4128194 | — | — | 1 | 9.72 |
| CHEMBL4130225 | — | — | 1 | 9.65 |
| CHEMBL4126027 | — | — | 1 | 8.94 |
| CHEMBL4128125 | — | — | 1 | 8.92 |
| CHEMBL4126738 | — | — | 1 | 8.69 |
| CHEMBL4126953 | — | — | 1 | 8.69 |
| CHEMBL4130148 | — | — | 1 | 6.94 |
| CHEMBL4130044 | — | — | 1 | 6.75 |
| CHEMBL4128112 | — | — | 1 | - |
| CHEMBL4524066 | — | — | 1 | - |
| CHEMBL4128276 | — | — | 1 | - |
| CHEMBL414357 | EXENATIDE | 4.0 | 1 | - |
| CHEMBL5314341 | GLUCAGON | 4.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4127525 | — | EC50 | = | 0.0397 | nM | 10.40 |
| CHEMBL4126812 | — | EC50 | = | 0.0582 | nM | 10.24 |
| CHEMBL4129347 | — | EC50 | = | 0.102 | nM | 9.99 |
| CHEMBL4128194 | — | EC50 | = | 0.189 | nM | 9.72 |
| CHEMBL4130225 | — | EC50 | = | 0.224 | nM | 9.65 |
| CHEMBL4126027 | — | EC50 | = | 1.16 | nM | 8.94 |
| CHEMBL4128125 | — | EC50 | = | 1.21 | nM | 8.92 |
| CHEMBL4126738 | — | EC50 | = | 2.032 | nM | 8.69 |
| CHEMBL4126953 | — | EC50 | = | 2.032 | nM | 8.69 |
| CHEMBL4130148 | — | EC50 | = | 114.0 | nM | 6.94 |
| CHEMBL4130044 | — | EC50 | = | 177.0 | nM | 6.75 |
| CHEMBL4128112 | — | EC50 | > | 1.0 | 10'8pM | - |
| CHEMBL4524066 | — | EC50 | > | 1.0 | 10'8pM | - |
| CHEMBL4128276 | — | EC50 | > | 1.0 | 10'8pM | - |
| CHEMBL414357 | EXENATIDE | EC50 | = | 2.0 | 10'5pM | - |
| CHEMBL5314341 | GLUCAGON | EC50 | > | 1.0 | 10'8pM | - |