Assay Detail
Functional
CHEMBL4135018
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against Bovine viral diarrhea virus NADL ATCC VR 534 infected in bovine MDBK cells assessed as protection against virus-induced cytopathic effect after 3 to 4 days by MTT assay
31
Total Activities
31
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Bovine viral diarrhea virus 1-NADL |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Target
Bovine viral diarrhea virus 1 (CHEMBL612571) ↗| Type | ORGANISM |
| Organism | Bovine viral diarrhea virus 1 |
Publication
Inhibitors of Yellow Fever Virus replication based on 1,3,5-triphenyl-4,5-dihydropyrazole scaffold: Design, synthesis and antiviral evaluation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 31 | 5.03 | 5.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4172978 | — | — | 1 | 5.60 |
| CHEMBL4169180 | — | — | 1 | 5.35 |
| CHEMBL4161254 | — | — | 1 | 5.26 |
| CHEMBL4165746 | — | — | 1 | 5.12 |
| CHEMBL4175245 | — | — | 1 | 5.00 |
| CHEMBL4177444 | — | — | 1 | 4.90 |
| CHEMBL1643 | RIBAVIRIN | 4.0 | 1 | 4.70 |
| CHEMBL4164614 | — | — | 1 | 4.28 |
| CHEMBL4174536 | — | — | 1 | - |
| CHEMBL1530025 | — | — | 1 | - |
| CHEMBL4166621 | — | — | 1 | - |
| CHEMBL4173042 | — | — | 1 | - |
| CHEMBL1881501 | — | — | 1 | - |
| CHEMBL1867917 | — | — | 1 | - |
| CHEMBL4168561 | — | — | 1 | - |
| CHEMBL4166223 | — | — | 1 | - |
| CHEMBL1591211 | — | — | 1 | - |
| CHEMBL1514645 | — | — | 1 | - |
| CHEMBL1441897 | — | — | 1 | - |
| CHEMBL4159714 | — | — | 1 | - |
| CHEMBL4170341 | — | — | 1 | - |
| CHEMBL1565276 | — | — | 1 | - |
| CHEMBL4173795 | — | — | 1 | - |
| CHEMBL4166525 | — | — | 1 | - |
| CHEMBL4177143 | — | — | 1 | - |
| CHEMBL4169949 | — | — | 1 | - |
| CHEMBL4162022 | — | — | 1 | - |
| CHEMBL4176360 | — | — | 1 | - |
| CHEMBL4169590 | — | — | 1 | - |
| CHEMBL4163087 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4172978 | — | EC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL4169180 | — | EC50 | = | 4500.0 | nM | 5.35 |
| CHEMBL4161254 | — | EC50 | = | 5500.0 | nM | 5.26 |
| CHEMBL4165746 | — | EC50 | = | 7500.0 | nM | 5.12 |
| CHEMBL4175245 | — | EC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL4177444 | — | EC50 | = | 12500.0 | nM | 4.90 |
| CHEMBL1643 | RIBAVIRIN | EC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL4164614 | — | EC50 | = | 52000.0 | nM | 4.28 |
| CHEMBL4166621 | — | EC50 | > | 36000.0 | nM | - |
| CHEMBL4169900 | — | EC50 | > | 19000.0 | nM | - |
| CHEMBL4173042 | — | EC50 | > | 5000.0 | nM | - |
| CHEMBL1881501 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1867917 | — | EC50 | > | 23000.0 | nM | - |
| CHEMBL4168561 | — | EC50 | > | 18000.0 | nM | - |
| CHEMBL4166223 | — | EC50 | > | 11000.0 | nM | - |
| CHEMBL1591211 | — | EC50 | > | 2000.0 | nM | - |
| CHEMBL1514645 | — | EC50 | > | 9000.0 | nM | - |
| CHEMBL1441897 | — | EC50 | > | 18000.0 | nM | - |
| CHEMBL1530025 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL4174536 | — | EC50 | > | 12000.0 | nM | - |
| CHEMBL4159714 | — | EC50 | > | 6000.0 | nM | - |
| CHEMBL4170341 | — | EC50 | > | 5000.0 | nM | - |
| CHEMBL1565276 | — | EC50 | > | 16000.0 | nM | - |
| CHEMBL4173795 | — | EC50 | > | 19000.0 | nM | - |
| CHEMBL4166525 | — | EC50 | > | 16000.0 | nM | - |
| CHEMBL4177143 | — | EC50 | > | 6000.0 | nM | - |
| CHEMBL4169949 | — | EC50 | > | 21000.0 | nM | - |
| CHEMBL4162022 | — | EC50 | > | 72000.0 | nM | - |
| CHEMBL4176360 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4169590 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4163087 | — | EC50 | > | 6000.0 | nM | - |