Assay Detail
Binding
CHEMBL4138803
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of L3MBTL1 (unknown origin) by AlphaScreen assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Lethal(3)malignant brain tumor-like protein 1 (CHEMBL1287622) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Methyllysine binding domains: Structural insight and small molecule probe development.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.78 | 7.01 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3351077 | CEFSULODIN | 2.0 | 1 | 7.01 |
| CHEMBL1257003 | — | — | 1 | 6.55 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3351077 | CEFSULODIN | IC50 | = | 98.0 | nM | 7.01 |
| CHEMBL1257003 | — | IC50 | = | 282.0 | nM | 6.55 |