Assay Detail
Binding
CHEMBL4139760
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of rat brain FAAH using [3H]AEA as substrate
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Novel propanamides as fatty acid amide hydrolase inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.21 | 5.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL191534 | — | — | 1 | 5.92 |
| CHEMBL1316 | CARPROFEN | 4.0 | 1 | 4.50 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL191534 | — | IC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL1316 | CARPROFEN | IC50 | = | 32000.0 | nM | 4.50 |