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Assay Detail

CHEMBL4146836

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured every minute for 10 mins by Ellman's method
59
Total Activities
55
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Acetylcholinesterase (CHEMBL220)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Novel donepezil-like N-benzylpyridinium salt derivatives as AChE inhibitors and their corresponding dihydropyridine "bio-oxidizable" prodrugs: Synthesis, biological evaluation and structure-activity relationship.
Azzouz R, Peauger L, Gembus V, Ţînţaş ML, Sopková-de Oliveira Santos J, Papamicaël C, Levacher V.
Eur J Med Chem (2018) 145 : 165 -190
PubMed 29324339 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 59 6.85 9.44

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4165327 1 9.44
CHEMBL4159705 1 8.57
CHEMBL4161065 1 8.00
CHEMBL4163678 1 7.96
CHEMBL4173239 1 7.78
CHEMBL4165973 1 7.74
CHEMBL4169938 1 7.68
CHEMBL4159880 1 7.65
CHEMBL4162015 1 7.62
CHEMBL4177133 1 7.53
CHEMBL4173784 1 7.43
CHEMBL4168037 1 7.37
CHEMBL4160115 1 7.26
CHEMBL4159243 1 7.16
CHEMBL4166513 1 7.15
CHEMBL4168987 1 6.96
CHEMBL4170331 1 6.93
CHEMBL4165562 1 6.84
CHEMBL4171568 1 6.77
CHEMBL4160696 4 6.76
CHEMBL4176179 1 6.68
CHEMBL4164981 1 6.62
CHEMBL4175003 1 6.56
CHEMBL4173405 1 6.51
CHEMBL4166464 1 6.42
CHEMBL4172353 1 6.25
CHEMBL4172797 1 6.25
CHEMBL4174372 1 6.05
CHEMBL4173313 1 6.05
CHEMBL4160310 1 6.04

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4165327 IC50 = 0.36 nM 9.44
CHEMBL4159705 IC50 = 2.7 nM 8.57
CHEMBL4161065 IC50 = 10.0 nM 8.00
CHEMBL4163678 IC50 = 11.0 nM 7.96
CHEMBL4173239 IC50 = 16.5 nM 7.78
CHEMBL4165973 IC50 = 18.1 nM 7.74
CHEMBL4169938 IC50 = 21.0 nM 7.68
CHEMBL4159880 IC50 = 22.2 nM 7.65
CHEMBL4162015 IC50 = 24.0 nM 7.62
CHEMBL4177133 IC50 = 29.5 nM 7.53
CHEMBL4173784 IC50 = 37.1 nM 7.43
CHEMBL4168037 IC50 = 43.0 nM 7.37
CHEMBL4160115 IC50 = 55.5 nM 7.26
CHEMBL4159243 IC50 = 69.3 nM 7.16
CHEMBL4166513 IC50 = 71.0 nM 7.15
CHEMBL4168987 IC50 = 110.5 nM 6.96
CHEMBL4170331 IC50 = 116.5 nM 6.93
CHEMBL4165562 IC50 = 143.5 nM 6.84
CHEMBL4171568 IC50 = 171.0 nM 6.77
CHEMBL4160696 IC50 = 173.0 nM 6.76
CHEMBL4176179 IC50 = 210.0 nM 6.68
CHEMBL4164981 IC50 = 242.4 nM 6.62
CHEMBL4175003 IC50 = 275.0 nM 6.56
CHEMBL4160696 IC50 = 286.0 nM 6.54
CHEMBL4173405 IC50 = 307.5 nM 6.51
CHEMBL4166464 IC50 = 378.8 nM 6.42
CHEMBL4160696 IC50 = 415.0 nM 6.38
CHEMBL4172353 IC50 = 568.0 nM 6.25
CHEMBL4172797 IC50 = 556.0 nM 6.25
CHEMBL4173313 IC50 = 896.0 nM 6.05
CHEMBL4174372 IC50 = 893.8 nM 6.05
CHEMBL4160310 IC50 = 923.0 nM 6.04
CHEMBL4160696 IC50 = 924.0 nM 6.03
CHEMBL4170940 IC50 = 1861.0 nM 5.73
CHEMBL4101303 IC50 = 5339.0 nM 5.27
CHEMBL4163016 IC50 = 9267.0 nM 5.03
CHEMBL4101303 IC50 = 26950.0 nM 4.57
CHEMBL4173562 IC50 > 10000.0 nM -
CHEMBL4174452 IC50 > 10000.0 nM -
CHEMBL4166141 IC50 > 10000.0 nM -
CHEMBL4174056 IC50 > 10000.0 nM -
CHEMBL4162692 IC50 > 10000.0 nM -
CHEMBL4170614 IC50 > 10000.0 nM -
CHEMBL4170921 IC50 > 10000.0 nM -
CHEMBL4172950 IC50 > 10000.0 nM -
CHEMBL4162281 IC50 > 10000.0 nM -
CHEMBL4175814 IC50 > 10000.0 nM -
CHEMBL4167954 IC50 > 10000.0 nM -
CHEMBL4167127 IC50 > 10000.0 nM -
CHEMBL4162993 IC50 > 10000.0 nM -