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Assay Detail

CHEMBL4147075

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Coxsackievirus B5 Ohio-1 ATCC VR 29 infected in African green monkey Vero 76 cells after 3 days by plaque reduction assay
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Coxsackievirus B5
Cell Type Vero 76
Confidence 1 — Organism
Curated By Intermediate

Target

Coxsackievirus B5 (CHEMBL613555)
Type ORGANISM
Organism Coxsackievirus B5

Publication

Quinoxaline derivatives as new inhibitors of coxsackievirus B5.
Carta A, Sanna G, Briguglio I, Madeddu S, Vitale G, Piras S, Corona P, Peana AT, Laurini E, Fermeglia M, Pricl S, Serra A, Carta E, Loddo R, Giliberti G.
Eur J Med Chem (2018) 145 : 559 -569
PubMed 29339251 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 10 6.46 8.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL29609 PLECONARIL 2.0 1 8.30
CHEMBL4171360 1 7.22
CHEMBL4163461 1 7.05
CHEMBL4168581 1 6.52
CHEMBL4160658 1 5.42
CHEMBL4165162 1 4.25
CHEMBL4170313 1 -
CHEMBL4159682 1 -
CHEMBL4173766 1 -
CHEMBL4163061 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL29609 PLECONARIL EC50 = 5.0 nM 8.30
CHEMBL4171360 EC50 = 60.0 nM 7.22
CHEMBL4163461 EC50 = 90.0 nM 7.05
CHEMBL4168581 EC50 = 300.0 nM 6.52
CHEMBL4160658 EC50 = 3800.0 nM 5.42
CHEMBL4165162 EC50 = 56000.0 nM 4.25
CHEMBL4170313 EC50 > 75000.0 nM -
CHEMBL4159682 EC50 > 100000.0 nM -
CHEMBL4173766 EC50 > 100000.0 nM -
CHEMBL4163061 EC50 > 100000.0 nM -