Assay Detail
Functional
CHEMBL4150993
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Growth inhibition of human MOLM13 cells after 4 days by WST-8 assay
17
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MOLM-13 |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Structure-Based Discovery of CF53 as a Potent and Orally Bioavailable Bromodomain and Extra-Terminal (BET) Bromodomain Inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 17 | 7.69 | 8.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4172447 | — | — | 1 | 8.30 |
| CHEMBL4166630 | — | — | 1 | 8.30 |
| CHEMBL4173488 | — | — | 1 | 8.15 |
| CHEMBL4172277 | — | — | 1 | 7.99 |
| CHEMBL4171109 | — | — | 1 | 7.97 |
| CHEMBL4161145 | — | — | 1 | 7.95 |
| CHEMBL4176849 | — | — | 1 | 7.93 |
| CHEMBL4174543 | — | — | 1 | 7.81 |
| CHEMBL4167996 | — | — | 1 | 7.75 |
| CHEMBL4162784 | — | — | 1 | 7.64 |
| CHEMBL4159422 | — | — | 1 | 7.58 |
| CHEMBL4175855 | — | — | 1 | 7.51 |
| CHEMBL4163185 | — | — | 1 | 7.41 |
| CHEMBL4169068 | — | — | 1 | 7.38 |
| CHEMBL4166235 | — | — | 1 | 7.25 |
| CHEMBL4170044 | — | — | 1 | 7.12 |
| CHEMBL4164563 | — | — | 1 | 6.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4172447 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL4166630 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL4173488 | — | IC50 | = | 7.0 | nM | 8.15 |
| CHEMBL4172277 | — | IC50 | = | 10.3 | nM | 7.99 |
| CHEMBL4171109 | — | IC50 | = | 10.6 | nM | 7.97 |
| CHEMBL4161145 | — | IC50 | = | 11.3 | nM | 7.95 |
| CHEMBL4176849 | — | IC50 | = | 11.7 | nM | 7.93 |
| CHEMBL4174543 | — | IC50 | = | 15.4 | nM | 7.81 |
| CHEMBL4167996 | — | IC50 | = | 17.7 | nM | 7.75 |
| CHEMBL4162784 | — | IC50 | = | 23.0 | nM | 7.64 |
| CHEMBL4159422 | — | IC50 | = | 26.6 | nM | 7.58 |
| CHEMBL4175855 | — | IC50 | = | 30.7 | nM | 7.51 |
| CHEMBL4163185 | — | IC50 | = | 38.8 | nM | 7.41 |
| CHEMBL4169068 | — | IC50 | = | 41.9 | nM | 7.38 |
| CHEMBL4166235 | — | IC50 | = | 56.0 | nM | 7.25 |
| CHEMBL4170044 | — | IC50 | = | 75.0 | nM | 7.12 |
| CHEMBL4164563 | — | IC50 | = | 201.0 | nM | 6.70 |