Assay Detail
Binding
CHEMBL4153978
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Inhibition of IL-5 in mouse Y16 cells assessed as reduction in cell proliferation after 48 hrs by WST-1 assay
44
Total Activities
44
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Identification of novel 2-benzyl-1-indanone analogs as interleukin-5 inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 44 | 4.83 | 5.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4176918 | — | — | 1 | 5.40 |
| CHEMBL1163396 | — | — | 1 | 5.30 |
| CHEMBL4169713 | — | — | 1 | 5.22 |
| CHEMBL4163488 | — | — | 1 | 4.77 |
| CHEMBL4173123 | — | — | 1 | 4.75 |
| CHEMBL4166938 | — | — | 1 | 4.69 |
| CHEMBL4165223 | — | — | 1 | 4.68 |
| CHEMBL4174194 | — | — | 1 | 4.61 |
| CHEMBL249466 | — | — | 1 | 4.58 |
| CHEMBL4169972 | — | — | 1 | 4.58 |
| CHEMBL4159659 | — | — | 1 | 4.55 |
| CHEMBL4161434 | — | — | 1 | - |
| CHEMBL4165925 | — | — | 1 | - |
| CHEMBL4176542 | — | — | 1 | - |
| CHEMBL4162488 | — | — | 1 | - |
| CHEMBL4173173 | — | — | 1 | - |
| CHEMBL4159098 | — | — | 1 | - |
| CHEMBL4169753 | — | — | 1 | - |
| CHEMBL4175849 | — | — | 1 | - |
| CHEMBL4171851 | — | — | 1 | - |
| CHEMBL4161793 | — | — | 1 | - |
| CHEMBL4166302 | — | — | 1 | - |
| CHEMBL4173558 | — | — | 1 | - |
| CHEMBL4162845 | — | — | 1 | - |
| CHEMBL4170104 | — | — | 1 | - |
| CHEMBL4159484 | — | — | 1 | - |
| CHEMBL4173792 | — | — | 1 | - |
| CHEMBL4165868 | — | — | 1 | - |
| CHEMBL4175242 | — | — | 1 | - |
| CHEMBL4159040 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4176918 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL1163396 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL4169713 | — | IC50 | = | 6000.0 | nM | 5.22 |
| CHEMBL4163488 | — | IC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL4173123 | — | IC50 | = | 18000.0 | nM | 4.75 |
| CHEMBL4166938 | — | IC50 | = | 20500.0 | nM | 4.69 |
| CHEMBL4165223 | — | IC50 | = | 21000.0 | nM | 4.68 |
| CHEMBL4174194 | — | IC50 | = | 24500.0 | nM | 4.61 |
| CHEMBL4169972 | — | IC50 | = | 26000.0 | nM | 4.58 |
| CHEMBL249466 | — | IC50 | = | 26200.0 | nM | 4.58 |
| CHEMBL4159659 | — | IC50 | = | 28000.0 | nM | 4.55 |
| CHEMBL4165925 | — | IC50 | - | — | - | |
| CHEMBL4167375 | — | IC50 | - | — | - | |
| CHEMBL4161434 | — | IC50 | - | — | - | |
| CHEMBL4169360 | — | IC50 | - | — | - | |
| CHEMBL4159248 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4169691 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4174244 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4159681 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4173967 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4162825 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4171974 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4159464 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4163933 | — | IC50 | - | — | - | |
| CHEMBL4174583 | — | IC50 | - | — | - | |
| CHEMBL4170769 | — | IC50 | - | — | - | |
| CHEMBL4160122 | — | IC50 | - | — | - | |
| CHEMBL4166302 | — | IC50 | - | — | - | |
| CHEMBL4159040 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4175242 | — | IC50 | - | — | - | |
| CHEMBL4165868 | — | IC50 | - | — | - | |
| CHEMBL4173792 | — | IC50 | - | — | - | |
| CHEMBL4159484 | — | IC50 | - | — | - | |
| CHEMBL4170104 | — | IC50 | - | — | - | |
| CHEMBL4162845 | — | IC50 | - | — | - | |
| CHEMBL4173558 | — | IC50 | - | — | - | |
| CHEMBL4176542 | — | IC50 | - | — | - | |
| CHEMBL4161793 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4171851 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4175849 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4169753 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4159098 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4173173 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4162488 | — | IC50 | > | 30000.0 | nM | - |