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Assay Detail

CHEMBL4190528

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HIV1 3B infected in human C8166 cells assessed as reduction in virus-induced cytopathic effect by measuring syncytium formation after 3 days by inverted microscopic analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human immunodeficiency virus 1
Cell Type C8166
Confidence 1 — Organism
Curated By Intermediate

Target

Human immunodeficiency virus 1 (CHEMBL378)
Type ORGANISM
Organism Human immunodeficiency virus 1

Publication

Chemical probes and inhibitors of bromodomains outside the BET family.
Moustakim M, Clark PGK, Hay DA, Dixon DJ, Brennan PE.
Medchemcomm (2016) 7 : 2246 -2264
PubMed 29170712 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 4.94 4.94

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4070058 1 4.94

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4070058 EC50 = 11520.0 nM 4.94