Assay Detail
Binding
CHEMBL4190560
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to ATAD2 (unknown origin) by isothermal titration calorimetry
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
ATPase family AAA domain-containing protein 2 (CHEMBL2150837) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Chemical probes and inhibitors of bromodomains outside the BET family.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 6.81 | 8.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4206758 | — | — | 1 | 8.10 |
| CHEMBL4216094 | — | — | 1 | 5.51 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4206758 | — | Kd | = | 8.0 | nM | 8.10 |
| CHEMBL4216094 | — | Kd | = | 3100.0 | nM | 5.51 |