Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL4190563

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to partial length human ATAD2B (Q955 to R1082) expressed in bacterial expression system by Bromoscan method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

ATPase family AAA domain-containing protein 2B (CHEMBL2176775)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Chemical probes and inhibitors of bromodomains outside the BET family.
Moustakim M, Clark PGK, Hay DA, Dixon DJ, Brennan PE.
Medchemcomm (2016) 7 : 2246 -2264
PubMed 29170712 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 9.00 9.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4206758 1 9.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4206758 Kd = 1.0 nM 9.00