Assay Detail
Binding
CHEMBL4195906
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human ERG by cell based automated patch clamp method
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Voltage-gated inwardly rectifying potassium channel KCNH2 (CHEMBL240) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Discovery of a Potent, Orally Bioavailable PI4KIIIβ Inhibitor (UCB9608) Able To Significantly Prolong Allogeneic Organ Engraftment in Vivo.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 20 | 5.24 | 5.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4210308 | — | — | 1 | 5.77 |
| CHEMBL4206816 | — | — | 1 | 5.70 |
| CHEMBL4205416 | — | — | 1 | 5.66 |
| CHEMBL4215244 | — | — | 1 | 5.10 |
| CHEMBL4203566 | — | — | 1 | 5.10 |
| CHEMBL4203041 | — | — | 1 | 4.77 |
| CHEMBL4217096 | — | — | 1 | 4.55 |
| CHEMBL4211181 | — | — | 1 | - |
| CHEMBL4209793 | — | — | 1 | - |
| CHEMBL1652677 | — | — | 1 | - |
| CHEMBL4207928 | — | — | 1 | - |
| CHEMBL4204100 | — | — | 1 | - |
| CHEMBL4208976 | — | — | 1 | - |
| CHEMBL4208440 | — | — | 1 | - |
| CHEMBL4213363 | — | — | 1 | - |
| CHEMBL4212822 | — | — | 1 | - |
| CHEMBL4217771 | — | — | 1 | - |
| CHEMBL4215340 | — | — | 1 | - |
| CHEMBL4204633 | — | — | 1 | - |
| CHEMBL4203671 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4210308 | — | IC50 | = | 1700.0 | nM | 5.77 |
| CHEMBL4206816 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL4205416 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL4215244 | — | IC50 | = | 8000.0 | nM | 5.10 |
| CHEMBL4203566 | — | IC50 | = | 8000.0 | nM | 5.10 |
| CHEMBL4203041 | — | IC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL4217096 | — | IC50 | = | 28000.0 | nM | 4.55 |
| CHEMBL4211181 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4209793 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL1652677 | — | IC50 | - | — | - | |
| CHEMBL4207928 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4204100 | — | IC50 | - | — | - | |
| CHEMBL4208976 | — | IC50 | - | — | - | |
| CHEMBL4208440 | — | IC50 | - | — | - | |
| CHEMBL4213363 | — | IC50 | - | — | - | |
| CHEMBL4212822 | — | IC50 | - | — | - | |
| CHEMBL4217771 | — | IC50 | - | — | - | |
| CHEMBL4215340 | — | IC50 | - | — | - | |
| CHEMBL4204633 | — | IC50 | - | — | - | |
| CHEMBL4203671 | — | IC50 | - | — | - |