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Assay Detail

CHEMBL4200980

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Functional
Antiviral activity against Dengue virus 1 Djibouti D1/H/IMTSSA/98/606 infected in African green monkey Vero cells assessed as reduction in viral yield after 7 days by qRT-PCR analysis
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism dengue virus type 1
Cell Type Vero
Confidence 1 — Organism
Curated By Intermediate

Target

dengue virus type 1 (CHEMBL613360)
Type ORGANISM
Organism dengue virus type 1

Publication

Discovery of Indole Derivatives as Novel and Potent Dengue Virus Inhibitors.
Bardiot D, Koukni M, Smets W, Carlens G, McNaughton M, Kaptein S, Dallmeier K, Chaltin P, Neyts J, Marchand A.
J Med Chem (2018) 61 : 8390 -8401
PubMed 30149709 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 6.63 7.33

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4212403 1 7.33
CHEMBL4205665 1 6.76
CHEMBL4215935 1 6.61
CHEMBL4212873 1 5.80

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4212403 EC50 = 47.0 nM 7.33
CHEMBL4205665 EC50 = 173.0 nM 6.76
CHEMBL4215935 EC50 = 247.0 nM 6.61
CHEMBL4212873 EC50 = 1600.0 nM 5.80