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Assay Detail

CHEMBL4234979

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Phototoxicity in HEK293 cells assessed as reduction in cell viability preincubated for 1 hr followed by LED light irradiation for 15 mins measured after 48 hrs by MTT assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HEK293
Confidence 1 — Organism
Curated By Intermediate

Target

HEK293 (CHEMBL614818)
Type CELL-LINE
Organism Homo sapiens

Publication

The design, synthesis, and evaluation of organic dithienopyrrole-based D-π-A dyes for use as sensitizers in photodynamic therapy.
Fuse S, Matsumura K, Takizawa M, Sato S, Nakamura H.
Bioorg Med Chem Lett (2018) 28 : 3099 -3104
PubMed 30055886 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 7.09 7.37

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4237757 1 7.37
CHEMBL3330737 1 6.80

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4237757 IC50 = 43.0 nM 7.37
CHEMBL3330737 IC50 = 160.0 nM 6.80