Assay Detail
Binding
CHEMBL4273591
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of PDE4C1 (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Intermediate |
Target
3',5'-cyclic-AMP phosphodiesterase 4C (CHEMBL291) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Lead-like Drugs: A Perspective.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.26 | 7.26 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL484785 | CRISABOROLE | 4.0 | 1 | 7.26 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL484785 | CRISABOROLE | IC50 | = | 55.0 | nM | 7.26 |