Assay Detail
Binding
CHEMBL4276646
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Binding affinity to human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysis
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Receptor-Ligand Interaction Measured by Inductively Coupled Plasma Mass Spectrometry and Selenium Labeling.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 3 | 9.28 | 9.49 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4278500 | — | — | 1 | 9.49 |
| CHEMBL4289837 | — | — | 1 | 9.35 |
| CHEMBL4294901 | — | — | 1 | 9.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4278500 | — | Kd | = | 0.32 | nM | 9.49 |
| CHEMBL4289837 | — | Kd | = | 0.45 | nM | 9.35 |
| CHEMBL4294901 | — | Kd | = | 0.99 | nM | 9.00 |