Assay Detail
Functional
CHEMBL4305663
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity against mouse 3T3 cells
21
Total Activities
21
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | NIH3T3 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Synthetic heterocyclic candidates as promising α-glucosidase inhibitors: An overview.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 21 | 6.21 | 6.21 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4468361 | — | — | 1 | 6.21 |
| CHEMBL4447393 | — | — | 1 | 6.21 |
| CHEMBL4475174 | — | — | 1 | 6.21 |
| CHEMBL4593619 | — | — | 1 | 6.21 |
| CHEMBL4435572 | — | — | 1 | 6.21 |
| CHEMBL4539228 | — | — | 1 | 6.21 |
| CHEMBL4455934 | — | — | 1 | 6.21 |
| CHEMBL4559950 | — | — | 1 | 6.21 |
| CHEMBL4456736 | — | — | 1 | 6.21 |
| CHEMBL4443159 | — | — | 1 | 6.21 |
| CHEMBL4513726 | — | — | 1 | 6.21 |
| CHEMBL4460638 | — | — | 1 | 6.21 |
| CHEMBL4548709 | — | — | 1 | 6.21 |
| CHEMBL4589941 | — | — | 1 | 6.21 |
| CHEMBL4567497 | — | — | 1 | 6.21 |
| CHEMBL4462006 | — | — | 1 | 6.21 |
| CHEMBL4550154 | — | — | 1 | 6.21 |
| CHEMBL4434647 | — | — | 1 | 6.21 |
| CHEMBL4465892 | — | — | 1 | 6.21 |
| CHEMBL4545512 | — | — | 1 | 6.21 |
| CHEMBL4593214 | — | — | 1 | 6.21 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4468361 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4447393 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4475174 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4593619 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4435572 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4539228 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4455934 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4559950 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4456736 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4443159 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4513726 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4460638 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4548709 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4589941 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4567497 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4462006 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4550154 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4434647 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4465892 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4545512 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL4593214 | — | IC50 | = | 610.0 | nM | 6.21 |