Assay Detail
Binding
CHEMBL4310225
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of recombinant His-tagged BRD9 (unknown origin) after 10 mins by TR-FRET assay
27
Total Activities
27
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
GNE-371, a Potent and Selective Chemical Probe for the Second Bromodomains of Human Transcription-Initiation-Factor TFIID Subunit 1 and Transcription-Initiation-Factor TFIID Subunit 1-like.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 27 | 5.82 | 6.64 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4436408 | — | — | 1 | 6.64 |
| CHEMBL4453202 | — | — | 1 | 6.21 |
| CHEMBL4513694 | — | — | 1 | 6.12 |
| CHEMBL4441257 | — | — | 1 | 6.07 |
| CHEMBL4448345 | — | — | 1 | 6.06 |
| CHEMBL4572531 | — | — | 1 | 6.05 |
| CHEMBL4470836 | — | — | 1 | 6.05 |
| CHEMBL4586175 | — | — | 1 | 6.02 |
| CHEMBL4483624 | — | — | 1 | 6.00 |
| CHEMBL4465624 | — | — | 1 | 6.00 |
| CHEMBL4436158 | — | — | 1 | 5.85 |
| CHEMBL4455513 | — | — | 1 | 5.85 |
| CHEMBL4520419 | — | — | 1 | 5.85 |
| CHEMBL4463398 | — | — | 1 | 5.82 |
| CHEMBL4483679 | — | — | 1 | 5.80 |
| CHEMBL4440829 | — | — | 1 | 5.80 |
| CHEMBL4566599 | — | — | 1 | 5.77 |
| CHEMBL4518929 | — | — | 1 | 5.77 |
| CHEMBL4466746 | — | — | 1 | 5.75 |
| CHEMBL4459660 | — | — | 1 | 5.70 |
| CHEMBL4459431 | — | — | 1 | 5.68 |
| CHEMBL4437997 | — | — | 1 | 5.66 |
| CHEMBL4468549 | — | — | 1 | 5.66 |
| CHEMBL4445482 | — | — | 1 | 5.62 |
| CHEMBL4448723 | — | — | 1 | 5.52 |
| CHEMBL4463538 | — | — | 1 | 5.02 |
| CHEMBL4534244 | — | — | 1 | 4.75 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4436408 | — | IC50 | = | 230.0 | nM | 6.64 |
| CHEMBL4453202 | — | IC50 | = | 620.0 | nM | 6.21 |
| CHEMBL4513694 | — | IC50 | = | 750.0 | nM | 6.12 |
| CHEMBL4441257 | — | IC50 | = | 860.0 | nM | 6.07 |
| CHEMBL4448345 | — | IC50 | = | 880.0 | nM | 6.06 |
| CHEMBL4572531 | — | IC50 | = | 900.0 | nM | 6.05 |
| CHEMBL4470836 | — | IC50 | = | 890.0 | nM | 6.05 |
| CHEMBL4586175 | — | IC50 | = | 960.0 | nM | 6.02 |
| CHEMBL4483624 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL4465624 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL4436158 | — | IC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL4455513 | — | IC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL4520419 | — | IC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL4463398 | — | IC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL4483679 | — | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL4440829 | — | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL4566599 | — | IC50 | = | 1700.0 | nM | 5.77 |
| CHEMBL4518929 | — | IC50 | = | 1700.0 | nM | 5.77 |
| CHEMBL4466746 | — | IC50 | = | 1800.0 | nM | 5.75 |
| CHEMBL4459660 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL4459431 | — | IC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL4437997 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL4468549 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL4445482 | — | IC50 | = | 2400.0 | nM | 5.62 |
| CHEMBL4448723 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL4463538 | — | IC50 | = | 9500.0 | nM | 5.02 |
| CHEMBL4534244 | — | IC50 | = | 18000.0 | nM | 4.75 |