Assay Detail
Functional
CHEMBL4316736
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Cytotoxicity against human HCT116 cells assessed as cell growth inhibition after 24 hrs by sulforhodamine B assay
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HCT-116 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
In Vitro and in Vivo Antitumor Effects of Plant-Derived Miliusanes and Their Induction of Cellular Senescence.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 15 | 5.32 | 5.71 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4513733 | — | — | 1 | 5.71 |
| CHEMBL4588940 | — | — | 1 | 5.59 |
| CHEMBL4572584 | — | — | 1 | 5.53 |
| CHEMBL4513721 | — | — | 1 | 5.46 |
| CHEMBL382849 | — | — | 1 | 5.43 |
| CHEMBL440759 | — | — | 1 | 5.41 |
| CHEMBL4515263 | — | — | 1 | 5.16 |
| CHEMBL4528773 | — | — | 1 | 5.14 |
| CHEMBL4458136 | — | — | 1 | 4.89 |
| CHEMBL4462375 | — | — | 1 | 4.85 |
| CHEMBL4520288 | — | — | 1 | - |
| CHEMBL4556341 | — | — | 1 | - |
| CHEMBL4579804 | — | — | 1 | - |
| CHEMBL4558393 | — | — | 1 | - |
| CHEMBL4544753 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4513733 | — | IC50 | = | 1950.0 | nM | 5.71 |
| CHEMBL4588940 | — | IC50 | = | 2570.0 | nM | 5.59 |
| CHEMBL4572584 | — | IC50 | = | 2930.0 | nM | 5.53 |
| CHEMBL4513721 | — | IC50 | = | 3430.0 | nM | 5.46 |
| CHEMBL382849 | — | IC50 | = | 3670.0 | nM | 5.43 |
| CHEMBL440759 | — | IC50 | = | 3940.0 | nM | 5.41 |
| CHEMBL4515263 | — | IC50 | = | 6970.0 | nM | 5.16 |
| CHEMBL4528773 | — | IC50 | = | 7180.0 | nM | 5.14 |
| CHEMBL4458136 | — | IC50 | = | 12900.0 | nM | 4.89 |
| CHEMBL4462375 | — | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL4520288 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4556341 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4579804 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4558393 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4544753 | — | IC50 | > | 30000.0 | nM | - |