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Assay Detail

CHEMBL4322376

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of FAAH (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Fatty-acid amide hydrolase 1 (CHEMBL2243)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

New Approaches to Cancer Therapy: Combining Fatty Acid Amide Hydrolase (FAAH) Inhibition with Peroxisome Proliferator-Activated Receptors (PPARs) Activation.
Brunetti L, Loiodice F, Piemontese L, Tortorella P, Laghezza A.
J Med Chem (2019) 62 : 10995 -11003
PubMed 31407888 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.25 5.25

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL191534 1 5.25

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL191534 IC50 = 5600.0 nM 5.25