Assay Detail
Functional
CHEMBL4329375
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Antiproliferative activity against human Kasumi-1 cells after 72 hrs by resazurin dye-based assay
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Kasumi 1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Highly fluorescent and HDAC6 selective scriptaid analogues.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 10 | 6.38 | 7.02 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4475116 | — | — | 1 | 7.02 |
| CHEMBL4526647 | — | — | 1 | 6.55 |
| CHEMBL4160632 | — | — | 1 | 6.54 |
| CHEMBL4461622 | — | — | 1 | 6.50 |
| CHEMBL4532304 | — | — | 1 | 6.44 |
| CHEMBL96051 | SCRIPTAID | — | 1 | 6.31 |
| CHEMBL4465218 | — | — | 1 | 6.24 |
| CHEMBL4476425 | — | — | 1 | 6.19 |
| CHEMBL4567832 | — | — | 1 | 6.09 |
| CHEMBL330201 | — | — | 1 | 5.96 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4475116 | — | IC50 | = | 96.0 | nM | 7.02 |
| CHEMBL4526647 | — | IC50 | = | 280.0 | nM | 6.55 |
| CHEMBL4160632 | — | IC50 | = | 290.0 | nM | 6.54 |
| CHEMBL4461622 | — | IC50 | = | 320.0 | nM | 6.50 |
| CHEMBL4532304 | — | IC50 | = | 360.0 | nM | 6.44 |
| CHEMBL96051 | SCRIPTAID | IC50 | = | 490.0 | nM | 6.31 |
| CHEMBL4465218 | — | IC50 | = | 570.0 | nM | 6.24 |
| CHEMBL4476425 | — | IC50 | = | 640.0 | nM | 6.19 |
| CHEMBL4567832 | — | IC50 | = | 810.0 | nM | 6.09 |
| CHEMBL330201 | — | IC50 | = | 1090.0 | nM | 5.96 |